Fragment-based approach applied to the discovery of protein-protein interactions stabilisers
Dario Valenti, Stanimira Hristeva, Christian Ottmann, Anna Karawajczyk
Taros
The next level in chemical space navigation: going far beyond enumerable compound libraries
Torsten Hoffmann, Marcus Gastreich
Drug Discov. Today, Mar. 2019, DOI:10.1016/j.drudis.2019.02.013;
Cardiomyocytes facing fibrotic conditions re-express extracellular matrix transcripts
Carlos O. Heras-Bautista, Nelly Mikhael, Jennifer Lam, Vaibhav Shinde, Alisa Katsen-Globa, Sabine Dieluweit, Marek Molcanyi, Vladimir Uvarov, Peter Jütten, Raja G.A. Sahito,…
Acta Biomater., Apr. 2019, 89, pp 180-192, DOI:10.1016/j.actbio.2019.03.017;
Cardiomyocytes facing fibrotic conditions re-express extracellular matrix transcripts Read More »
Clinical candidates modulating protein-protein interactions: The fragment-based experience
Dario Valenti, Stanimira Hristeva, Dimitrios Tzalis, and Christian Ottmann
Eur. J. Med. Chem., Apr. 2019, 167, pp 76-95, DOI: 10.1016/j.ejmech.2019.01.084;
DPD-Inspired Discovery of Novel LsrK Kinase Inhibitors: An Opportunity To Fight Antimicrobial Resistance
Silvia Stotani, Viviana Gatta, Prasanthi Medarametla, Mohan Padmanaban, Anna Karawajczyk, Fabrizio Giordanetto, Päivi Tammela,…
J. Med. Chem., Feb. 2019, DOI: 10.1021/acs.jmedchem.9b00025;
Screening of Novel Feruloyl Esterases from Talaromyces Wortmannii for the Development of Efficient and Sustainable Syntheses of Feruloyl Derivatives
Io Antonopoulou, Laura Iancu, Peter Jütten, Alexander Piechot,…
Enzyme Microb. Technol., Jan. 2019, 120, pp 124–135., DOI:10.1016/j.enzmictec.2018.08.007.;
Optimization of Enzymatic Synthesis of L-Arabinose Ferulate Catalyzed by Feruloyl Esterases from Myceliophthora Thermophila
Io Antonopoulou, Adamantia Papadopoulou, Laura Iancu, Gabriella Cerullo, Marianna Ralli, Peter Jütten,…
Process Biochemistry, Nov. 2017, 65, pp 100–108., DOI:10.1016/j.procbio.2017.11.009.;
Targeted Stabilizers of Protein-Protein Interactions as a Novel Class of Therapeutic Agents and Basic Research Tool Compounds
Dario Valenti, Stanimira Hristeva, Anna Karawajczyk, Dimitrios Tzalis
Taros, TASPPI
A Versatile Strategy for the Synthesis of 4,5-Dihydroxy-2,3-Pentanedione (DPD) and Related Compounds as Potential Modulators of Bacterial Quorum Sensing
Silvia Stotani, Viviana Gatta, Federico Medda, Mohan Padmanaban, Anna Karawajczyk, Päivi Tammela, Fabrizio Giordanetto, Dimitrios Tzalis and Simona Collina
Molecules 2018, 23, 2545
Optimization of Transesterification Reactions with CLEA-Immobilized Feruloyl Esterases
Anastasia Zerva, Io Antonopoulou, Josefine Enman, Laura Iancu, Peter Jütten,…
Molecules, Sept. 2018, 23, 2403., DOI:10.3390/molecules23092403.;
Optimization of Transesterification Reactions with CLEA-Immobilized Feruloyl Esterases Read More »